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yzshua1987金蟲 (正式寫手)
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[求助]
求翻譯一段話,藥理專業(yè)的進(jìn)
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| Contemporary receptor theory was developed to account for the existence of constitutive activity, as defined by the presence of receptor signaling in the absence of any ligand. Thus, ligands acting at a constitutively active receptor, can act as agonists, antagonists, and inverse agonists.In vitro studies have also revealed the complexity of ligand/receptor interactions including agonist-directed stimulus trafficking, a finding that has led to multi-active state models of receptor function. 重點是翻譯紅色部分,這幾個詞遇到很多次了,不太理解,能解釋下意思更好,謝謝了 |

金蟲 (著名寫手)

新蟲 (初入文壇)
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“隨著在沒有任何配基的情況下受體信號存在的確定,當(dāng)代受體理論被認(rèn)為是構(gòu)效關(guān)系存在的原因所在。因此,配基對結(jié)構(gòu)性效應(yīng)的受體起作用,可作為激動劑,拮抗劑,或反激動劑。另外,體外研究也揭示了配體/受體的相互作用的復(fù)雜性,包括激動劑定向刺激因子,一項導(dǎo)致受體功能多活性模型的發(fā)現(xiàn)! 我能力有限,僅供參考啊 ………… |
金蟲 (正式寫手)

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