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[求助]
急急急,他克莫司的理化性質(zhì)參數(shù)?
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| 我現(xiàn)在急要他克莫司的理化性質(zhì)參數(shù)的數(shù)據(jù),包括脂水分配系數(shù),通透性,pKa,溶解度,血漿蛋白結(jié)合率,全血血漿分配比,這些性質(zhì)的具體的數(shù)值在哪里可以找到。空(qǐng)高人指點(diǎn)下啊。謝謝了! |


版主 (文壇精英)
老痞
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Pharmaprojects數(shù)據(jù)庫(kù),或化學(xué)物質(zhì)索引數(shù)據(jù)庫(kù)http://www.drugfuture.com/chemdata/ 該化合物專(zhuān)利EP184162。 化學(xué)物質(zhì)索引數(shù)據(jù)庫(kù) Properties: Colorless prisms from acetonitrile, mp 127-129°. [a]D23 -84.4° (c = 1.02 in chloroform). Sol in methanol, ethanol, acetone, ethyl acetate, chloroform, diethyl ether; sparingly sol in hexane, petroleum ether. Insol in water. LD50 i.p. in mice: >200 mg/kg (Kino). LD50 in male, female rats (mg/kg): 57.0, 23.6 i.v.; 134, 194 orally (Ohara). |

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