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[求助]
藥化專利 摘要翻譯 漢譯英 急
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發(fā)明名稱:新的喹啉類化合物及其用途 發(fā)明書摘要 本發(fā)明涉及通式Ⅰ所示的喹啉類衍生物與其幾何異構(gòu)體及它們藥學(xué)上可接受的鹽、水合物或前藥,其中取代基M、R1、R2、X、Y具有在說明書中給出的含義。本發(fā)明還涉及通式Ⅰ的化合物具有強(qiáng)的抑制c-Met激酶的作用,并且還涉及該類化合物及其藥學(xué)上可接受的鹽、水合物在制備治療由于c-Met激酶異常高表達(dá)所引起疾病的藥物中的用途,特別是在制備治療和/或預(yù)防癌癥的藥物中的用途。 |
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Title:Quinoline derivatives and uses thereof Abstract The present invention relates to quinoline derivatives of formula I, optical isomers, pharmaceutically acceptable salts, hydrates and/or prodrug thereof. Wherein: substituents M, R1, R2, X, and Y are as defined in the description. The present invention also relates to compounds of formula I, their pharmaceutically acceptable salts and/or hydrates, which have potent inhibitory effect of c-Met kinase, can be used in preparation for treating the abnormal c-Met kinase overexpression-related diseases, especially for preparation of treatment and/or prevention of cancer. |
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