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名我天下木蟲 (正式寫手)
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| 作為目前應(yīng)用最廣泛的體外吸收模型, Caco- 2 細(xì)胞模型能夠在分子水平預(yù)測藥物的吸收、轉(zhuǎn)運(yùn)特征, 并能夠研究藥物之間的相互作用。國內(nèi)外已經(jīng)有人將Caco- 2 細(xì)胞模型用于天然藥物研究, 熱點(diǎn)集中在黃酮類、生物堿類和皂苷類物質(zhì), 應(yīng)用最多的是藥物代謝和生物利用度研究, 另外還有用于觀察單一成分的藥理活性和藥物胃腸毒性的報道 |

| As the most widely used absorption model in vitro presently,Caco- 2 cell model can estimate drug absorption,transport characteristics at molecular level and study the interactions among drugs. Caco - 2 cell model has been used for natural medicine research, which was concentrated on flavonoids, alkaloids and saponins , be used for drug metabolism and bioavailability mostly and employed to observe pharmacological activity of single constituents and gastrointestinal toxicity. |
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