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In mice, mortality, severity and incidence of neurotoxicity and leukopenia occurred at cumulative dose levels which were comparable to the corresponding single-dose levels , e .g. the cumulative 5-day LD50 was 450 mg/ m2(5x 90 mg m2) which correlates well with the single-dose LD50 of 414 mg/ m2. In dogs, gastrointestinal toxicity and leukopenia of cumulative daily doses were of a severity corresponding to comparable single-dose levels: five daily doses of 6 mg/m2 produced adverse effects comparable to those following a single dose of 30 mg/m2. |

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| 在小鼠,累積劑量引起的死亡率,神經(jīng)毒性嚴(yán)重程度和白細(xì)胞減少癥的發(fā)病率與單一劑量水平相近,例如,累積5天的LD50(半數(shù)致死量)為450毫克/米2(5×90毫克/平方米),與單一劑量半數(shù)致死量414毫克/米2有良好的相關(guān)性。在狗,累積每日劑量引起胃腸道毒性和白細(xì)胞減少癥與單一劑量引起的嚴(yán)重程度相當(dāng):5天每日劑量為6毫克/平方米引起的副作用和單一劑量30mg/m2相仿。 |
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